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    Discovery and optimization of wt-RET/KDR-selective inhibitors of RET(V804M) kinase

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    Authors
    Newton, Rebecca
    Waszkowycz, Bohdan
    Seewooruthun, C
    Burschowsky, D
    Richards, M
    Hitchin, Samantha
    Begum, Habiba
    Watson, Amanda J
    French, Eleanor
    Hamilton, Niall M
    Jones, Stuart
    Lin, LY
    Waddell, Ian D
    Echalier, A
    Bayliss, R
    Jordan, Allan M
    Ogilvie, Donald J
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    Affiliation
    Drug Discovery Unit, Cancer Research UK, Manchester Institute, University of Manchester, Alderley Park, Macclesfield SK10 4TG, U.K.
    Issue Date
    2020
    
    Metadata
    Show full item record
    Citation
    Newton R, Waszkowycz B, Seewooruthun C, Burschowsky D, Richards M, Hitchin S, et al. Discovery and Optimization of wt-RET/KDR-Selective Inhibitors of RET(V804M) Kinase. ACS Med Chem Lett. 2020;11(4):497-505.
    Journal
    ACS Medicinal Chemistry Letters
    URI
    http://hdl.handle.net/10541/622991
    DOI
    10.1021/acsmedchemlett.9b00615
    PubMed ID
    32292556
    Additional Links
    https://dx.doi.org/ 10.1021/acsmedchemlett.9b00615
    Type
    Article
    Language
    en
    ae974a485f413a2113503eed53cd6c53
    10.1021/acsmedchemlett.9b00615
    Scopus Count
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